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Table 1 List of 32 tested protein kinases for in vitro enzymatic profiling.

From: Homopharma: A new concept for exploring the molecular binding mechanisms and drug repurposing

Sequence group

Symbol name

Kinase SK number

Kinase description

AKT2

AGC

SK019

v-akt murine thymoma viral oncogene homolog 2

DMPK

AGC

SK111

dystrophia myotonica-protein kinase

PRKCA

AGC

SK303

protein kinase C, alpha

RPS6KA1

AGC

SK338

ribosomal protein S6 kinase, 90kDa, polypeptide 1

CAMK2G

CAMK

SK060

calcium/calmodulin-dependent protein kinase (CaM kinase) II gamma

CAMK4

CAMK

SK061

calcium/calmodulin-dependent protein kinase IV

CHEK1

CAMK

SK078

CHK1 checkpoint homolog (S. pombe)

CHEK2

CAMK

SK079

CHK2 checkpoint homolog (S. pombe)

PIM1

CAMK

SK291

pim-1 oncogene

CSNK1G1

CK1

SK647

casein kinase 1, gamma 1

VRK1

CK1

SK389

vaccinia related kinase 1

CDK6

CMGC

SK071

cyclin-dependent kinase 6

CLK3

CMGC

SK092

CDC-like kinase 3

CSNK2A1

CMGC

SK088

casein kinase 2, alpha 1 polypeptide

MAPK10

CMGC

SK190

mitogen-activated protein kinase 10

MAPK14

CMGC

SK264

mitogen-activated protein kinase 14

MAPK3

CMGC

SK134

mitogen-activated protein kinase 3

MAP2K1

STE

SK217

mitogen-activated protein kinase kinase 1

STK10

STE

SK426

serine/threonine kinase 10

STK24

STE

SK246

serine/threonine kinase 24 (STE20 homolog, yeast)

EGFR

TK

SK118

epidermal growth factor receptor (erythroblastic leukemia viral (v-erb-b) oncogene homolog, avian)

FGFR1

TK

SK143

fibroblast growth factor receptor 1 (fms-related tyrosine kinase 2, Pfeiffer syndrome)

IGF1R

TK

SK174

insulin-like growth factor 1 receptor

INSR

TK

SK178

insulin receptor

KIT

TK

SK201

v-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog

LCK

TK

SK206

lymphocyte-specific protein tyrosine kinase

SRC

TK

SK357

v-src sarcoma (Schmidt-Ruppin A-2) viral oncogene homolog (avian)

SYK

TK

SK363

spleen tyrosine kinase

ACVR1

TKL

SK026

activin A receptor, type I

LIMK1

TKL

SK412

LIM domain kinase 1

MAP3K7

TKL

SK364

mitogen-activated protein kinase kinase kinase 7

RAF1

TKL

SK324

v-raf-1 murine leukemia viral oncogene homolog 1